孙培培教授课题组在JOURNAL OF ORGANIC CHEMISTRY发表研究论文

时间:2019-11-11 来源:化科院 点击数:

TBHP/KI-Promoted Annulation of Anilines, Ethers, and Elemental Sulfur: Access to 2-Aryl-, 2-Heteroaryl-, or 2-Alkyl-Substituted Benzothiazoles
Zhang, J (Zhang, Jie)[ 1 ] ; Zhao, X (Zhao, Xin)[ 1 ] ; Liu, P (Liu, Ping)[ 1 ]*(刘平); Sun, PP (Sun, Peipei)[ 1 ]*(孙培培)

[ 1 ] Nanjing Normal Univ, Jiangsu Collaborat Innovat Ctr Biomed Funct Mat, Sch Chem & Mat Sci, Jiangsu Prov Key Lab Mat Cycle Proc & Pollut Cont, Nanjing 210023, Jiangsu, Peoples R China

JOURNAL OF ORGANIC CHEMISTRY,201910,84(19),12596-12605

An efficient TBHP/KI-promoted annulation of anilines with ethers and elemental sulfur has been developed through the selective C-O bond cleavage of ethers under transition-metal-free conditions. A wide range of 2-aryl-, 2-heteroaryl-, and 2-alkyl-substituted benzothiazoles were easily prepared with satisfactory yields and good functional group compatibility.

文章链接:
https://pubs.acs.org/doi/10.1021/acs.joc.9b02145

Copyright © 2009-20010 南京师范大学 化学与材料科学学院. All rights reserved.